The 5-HT3 receptor belongs to the Cys-loop superfamily of ligand-gated ion channels (LGICs) and therefore differs structurally and functionally from all...
22 KB (2,395 words) - 18:29, 18 July 2024
The 5-HT3 antagonists, informally known as "setrons", are a class of drugs that act as receptor antagonists at the 5-HT3 receptor, a subtype of serotonin...
43 KB (4,628 words) - 10:52, 21 February 2024
response. The exception to this is the 5-HT3 receptor which is a ligand-gated ion channel. In 2014, a novel 5-HT receptor was isolated from the small white butterfly...
65 KB (5,263 words) - 10:40, 12 August 2024
Ondansetron (category 5-HT3 antagonists)
It is a serotonin 5-HT3 receptor antagonist. It does not have any effect on dopamine receptors or muscarinic acetylcholine receptors. Ondansetron was patented...
34 KB (3,154 words) - 19:29, 13 July 2024
5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
2 KB (166 words) - 00:47, 13 May 2022
subclass consists of drugs selectively acting at the 5-HT3 receptors, and thus are known as 5-HT3 antagonists. They are efficacious in treating chemotherapy-induced...
5 KB (506 words) - 03:46, 13 August 2023
sickness and the more serious hyperemesis gravidarum. 5-HT3 receptor antagonists block serotonin receptors in the central nervous system and gastrointestinal...
16 KB (1,680 words) - 19:38, 18 August 2024
individuals. 2-Methyl-5-hydroxytryptamine (2-methylserotonin) and quipazine are moderately selective agonists of the 5-HT3 receptor that are used in scientific...
16 KB (1,657 words) - 17:23, 8 June 2024
D2 receptors, serotonin 5-HT3 receptors, opioid receptors, acetylcholine receptors, and receptors for substance P. Stimulation of different receptors are...
22 KB (2,404 words) - 02:48, 4 September 2023
Vortioxetine (category 5-HT3 antagonists)
the serotonin 5-HT1A receptor, partial agonist of the 5-HT1B receptor, and antagonist of the serotonin 5-HT1D, 5-HT3, and 5-HT7 receptors, as well as an...
56 KB (4,803 words) - 19:52, 31 August 2024