Bosentan, sold under the brand name Tracleer among others, is a dual endothelin receptor antagonist medication used in the treatment of pulmonary artery...
13 KB (1,113 words) - 16:17, 2 May 2024
which affect both endothelin A (ETA) and B receptors (ETB) aprocitentan, bosentan, macitentan, tezosentan Selective ETA Receptor Antagonists, which affect...
1 KB (108 words) - 13:59, 11 July 2024
arterial hypertension (PAH). The other two ERAs marketed as of 2014 are bosentan and ambrisentan. Macitentan is a dual ERA, meaning that it acts as an antagonist...
11 KB (1,028 words) - 01:35, 6 May 2024
(COX-2 inhibitor) Celecoxib (COX-2 inhibitor) Parecoxib (COX-2 inhibitor) Bosentan (endothelin receptor antagonist) Dofetilide (class III antiarrhythmic)...
4 KB (260 words) - 08:48, 25 November 2023
treat pulmonary hypertension include epoprostenol, treprostinil, iloprost, bosentan, ambrisentan, macitentan, and sildenafil, tadalafil, selexipag, riociguat...
89 KB (8,893 words) - 16:41, 6 July 2024
pulmonary hypertension, which was treatable in preliminary research by bosentan, sitaxentan or ambrisentan. Endothelins have involvement in cardiovascular...
17 KB (1,655 words) - 20:05, 8 December 2023
Examples of such sodium salts are (selection): Bispyribac, bithionol, bosentan, brequinar, bromfenac, Cefmenoxime, ceftiofur, citicoline, diclofenac ...
3 KB (314 words) - 18:14, 20 April 2023
prostacyclin analogue iloprost, and the dual endothelin-receptor antagonist bosentan may be beneficial for Raynaud's phenomenon. Skin tightness may be treated...
40 KB (4,696 words) - 14:56, 12 June 2024
same as bosentan, but the hepatotoxicity of sitaxentan outweighs its benefits. Dosing is once daily, as opposed to twice daily for bosentan. On December...
8 KB (711 words) - 22:23, 21 March 2024
inhibitors (e.g., sildenafil) or iloprost Prevention of new digital ulcers with bosentan Malnutrition, secondary to intestinal flora overgrowth with tetracycline...
38 KB (3,291 words) - 01:18, 9 May 2024